Authors

  • M.O.Shomaksudova
    Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of The Republic Of Uzbekistan
  • A.A.Tulaganov
    Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of The Republic Of Uzbekistan
  • A.D.Matchanov
    Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of The Republic Of Uzbekistan
  • D.M.Sarvarova
    Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of The Republic Of Uzbekistan

DOI:

https://doi.org/10.37547/ajbspi/Volume04Issue01-17

Keywords:

Dry extract saffron chromatography

Abstract

The article presents the results of a study of biologically active substances in a dry extract obtained from the flower buds of the medicinal plant saffron Crocus sativus L. The GSX method was developed to determine the amount of biologically active substances in the dry extract.


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Volume 04 Issue 01-2024

113


American Journal Of Biomedical Science & Pharmaceutical Innovation
(ISSN

2771-2753)

VOLUME

04

ISSUE

01

P

AGES

:

113-117

SJIF

I

MPACT

FACTOR

(2021:

5.

705

)

(2022:

5.

705

)

(2023:

6.534

)

OCLC

1121105677















































Publisher:

Oscar Publishing Services

Servi

ABSTRACT

The article presents the results of a study of biologically active substances in a dry extract obtained from the flower

buds of the medicinal plant saffron Crocus sativus L. The GSX method was developed to determine the amount of

biologically active substances in the dry extract.

KEYWORDS

Dry extract, saffron, chromatography, standard samples.

INTRODUCTION

Research Article

QUANTITATIVE

DETERMINATION

OF

BIOLOGICALLY

ACTIVE

COMPOUNDS FROM DRY EXTRACT OF SAFFRON (CROCUS SATIVUS L.)
BY GAS CHROMATOGRAPHY

Submission Date:

January 21, 2024,

Accepted Date:

January 26, 2024,

Published Date:

January 31, 2024

Crossref doi:

https://doi.org/10.37547/ajbspi/Volume04Issue01-17


M.O.Shomaksudova

Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of
The Republic Of Uzbekistan

A.A.Tulaganov

Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of
The Republic Of Uzbekistan

A.D.Matchanov

Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of
The Republic Of Uzbekistan

D.M.Sarvarova

Tashkent Pharmaceutical Institute, Uzkfiti, Institute Of Bioorganic Chemistry Of The Academy Of Sciences Of
The Republic Of Uzbekistan

Journal

Website:

https://theusajournals.
com/index.php/ajbspi

Copyright:

Original

content from this work
may be used under the
terms of the creative
commons

attributes

4.0 licence.


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Volume 04 Issue 01-2024

114


American Journal Of Biomedical Science & Pharmaceutical Innovation
(ISSN

2771-2753)

VOLUME

04

ISSUE

01

P

AGES

:

113-117

SJIF

I

MPACT

FACTOR

(2021:

5.

705

)

(2022:

5.

705

)

(2023:

6.534

)

OCLC

1121105677















































Publisher:

Oscar Publishing Services

Servi

Chromatography makes it possible to carry out

qualitative and quantitative analysis of the objects

under study, study the physical and chemical

properties of substances, and monitor and

automatically regulate technological processes. Gas

chromatography is a method for separating volatile

compounds.

This method can analyze gaseous, liquid and solid

substances with a molecular weight of less than 400

that satisfy certain requirements, the main ones being

volatility, thermal stability, inertness and ease of

preparation. Quantitative analysis can only be carried

out if the substance is heat-resistant, i.e. evaporates

reproducibly in the dispenser and elutes from the

column without decomposition (1,7).

In pharmaceutical analysis, the GLC method is

widely used to determine residual organic solvents in

pharmaceutical

substances,

biological

active

substances in liquid and dry extracts of medicinal plant

materials, as well as in assessing the quality of essential

oils, volatile medicinal substances, and their

preparations (2,5,6).

The purpose of our work is to study the

quantitative content of biological active substances in

a dry extract obtained from plant raw materials of

saffron using gas-liquid chromatography. Previously,

we studied the qualitative content of biologically active

substances in plant raw materials of saffron using gas

chromatography-mass spectroscopy (3).

For the quantitative determination of

biologically active substances in the dry extract of

saffron, we used the dry extract we had previously

obtained by the percolation method (4).

Experimental parts.

Quantification method:

Gas chromatograph

Khromatek-Kristall

5000 (Russia)

Detector-FID

Detector temperature

250 0С

Thermostat temperature (gradient) -

70 0С (6min), 1500С (6

-

15min), 200 0С (15

-

33min), 220 0С (33

-38min)

Injector temperature -

200 0С

Carrier gas

nitrogen

Split flow

1/20

Injection

1 µl


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Volume 04 Issue 01-2024

115


American Journal Of Biomedical Science & Pharmaceutical Innovation
(ISSN

2771-2753)

VOLUME

04

ISSUE

01

P

AGES

:

113-117

SJIF

I

MPACT

FACTOR

(2021:

5.

705

)

(2022:

5.

705

)

(2023:

6.534

)

OCLC

1121105677















































Publisher:

Oscar Publishing Services

Servi

Fig. 1 Chromatogram of standard samples

Figure 1 shows chromatogram data for the three main standard substances isophorone with a retention time of 26.777

min, 2,6,6-trimethylcyclohexa-1,3-diene-1-carbaldehyde with a column retention time of 28.783 min, and 4-

ochophorone with a retention time of 30.916 min . For comparison, the concentration of standard samples was 3

mg/ml.

Fig 2 Chromatogram of hexane extract of dry extract of Saffron


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Volume 04 Issue 01-2024

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American Journal Of Biomedical Science & Pharmaceutical Innovation
(ISSN

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VOLUME

04

ISSUE

01

P

AGES

:

113-117

SJIF

I

MPACT

FACTOR

(2021:

5.

705

)

(2022:

5.

705

)

(2023:

6.534

)

OCLC

1121105677















































Publisher:

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From the data presented in Fig. 2, it is clear that in the hexane extract of the Saffron plant all three main components

are observed: isophorone with a retention time of 26.766 minutes, 2,6,6-trimethylcyclohexa-1,3-dien-1-carbaldehyde

with a retention time of column 28.751 min and 4-ochophorone with a retention time of 30.875 min. The quantitative

content of isophorone is 0.76 mg/ml, 2,6,6-trimethylcyclohexa-1,3-diene-1-carbaldehyde is 5.71 mg/ml and 4-

ochophorone is 0.68 mg/ml.

Fig 3 Chromatogram of acetonitrile extract of dry extract of Saffron

From the data presented in Fig. 3, it is clear that in the

acetonite extract of the Saffron plant two main

components are observed: 2,6,6-trimethylcyclohexa-

1,3-diene-1-carbaldehyde with a retention time on the

column of 28.745 minutes and 4-ochophorone with

retention time 30.877 min. The quantitative content of

2,6,6-trimethylcyclohexa-1,3-diene-1-carbaldehyde

is

0.44 mg/ml and 4-ochophorone is 0.42 mg/ml.

Conclusion. Thus, studies have shown that for the

extraction of Saffron it is relatively more effective to

use hexane as a solvent.

REFERENCES

1.

Е.А. Кривошеев, Р.И. Саяхов. «Газовая

хроматография» Методические указания к

лабораторной работе Казань, 2021. 23 с. ВВ.

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В.

Тыжигирова

«Газовая

хроматография»Краткая

характеристика

метода

и

его

применение

в

фармацевтическом

анализе

Учебное

пособие Иркутск ИГМУ 2016

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М.О.

Шомахсудова,

А.А.

Тулаганов,

Я.К.Назирова, С.З. Нишанбаев. «Разработка


background image

Volume 04 Issue 01-2024

117


American Journal Of Biomedical Science & Pharmaceutical Innovation
(ISSN

2771-2753)

VOLUME

04

ISSUE

01

P

AGES

:

113-117

SJIF

I

MPACT

FACTOR

(2021:

5.

705

)

(2022:

5.

705

)

(2023:

6.534

)

OCLC

1121105677















































Publisher:

Oscar Publishing Services

Servi

методов анализа биологически актывних

веществ в растительном сыре шафрана

посевного(Crocus sativus L) с помощью

хромато

-

спектрометрии»,

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практической

конференции. “Современная фармация

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исследования ”,приуроченной к 20

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летию

факультета Фармация. 5май 2022й Нур

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Султан.

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Zuparova, Z. A., Olimov, N. K., Ismoilova, G. M.,

& Khasanova, B. J. (2020). Determination of

high quality of echinaceae purpurae herba

grown in Uzbekistan and the prospect of

creating

immunomodulatory

medicinal

products on its base. International Journal of

Psychosocial Rehabilitation, 24(4), 2355-2366.

6.

Zuparova, Z. A., and G. M. Ismoilova.

"Determining The Authenticity Of Immunacea

Bio Tablets With Immunomodulatory Action."

Journal of Pharmaceutical Negative Results

(2022): 2637-2641.

7.

Sarvarova, D. M., et al. "Study Of The

Assortment Of Antioxidant And Hemostatic

Medicines Registered In The Republic Of

Uzbekistan."

Journal of

Pharmaceutical

Negative Results (2023): 1028-1033.

References

Е.А. Кривошеев, Р.И. Саяхов. «Газовая хроматография» Методические указания к лабораторной работе Казань, 2021. 23 с. ВВ.

В. Тыжигирова «Газовая хроматография»Краткая характеристика метода и его применение в фармацевтическом анализе Учебное пособие Иркутск ИГМУ 2016

М.О. Шомахсудова, А.А. Тулаганов, Я.К.Назирова, С.З. Нишанбаев. «Разработка методов анализа биологически актывних веществ в растительном сыре шафрана посевного(Crocus sativus L) с помощью хромато-спектрометрии», Pharmaceutical journal, №2, том.29, 2020 Тошкент.

Шомаксудова М.О., Тулаганов А.А. .XI Международной научно-практической конференции. “Современная фармация новые падходы в образовании актуальные исследования ”,приуроченной к 20-летию факультета Фармация. 5май 2022й Нур-Султан.

Zuparova, Z. A., Olimov, N. K., Ismoilova, G. M., & Khasanova, B. J. (2020). Determination of high quality of echinaceae purpurae herba grown in Uzbekistan and the prospect of creating immunomodulatory medicinal products on its base. International Journal of Psychosocial Rehabilitation, 24(4), 2355-2366.

Zuparova, Z. A., and G. M. Ismoilova. "Determining The Authenticity Of Immunacea Bio Tablets With Immunomodulatory Action." Journal of Pharmaceutical Negative Results (2022): 2637-2641.

Sarvarova, D. M., et al. "Study Of The Assortment Of Antioxidant And Hemostatic Medicines Registered In The Republic Of Uzbekistan." Journal of Pharmaceutical Negative Results (2023): 1028-1033.