Authors

  • Oyjamol Uzoqova
  • Nilufar Boboqulova
  • Farida Axsanova

DOI:

https://doi.org/10.71337/inlibrary.uz.science-research.71937

Abstract

Many RCTs have shown that monotherapy reduces blood pressure only in a limited number of hypertension cases, and most patients require a combination of at least two drugs for satisfactory blood pressure control. A meta-analysis of more than 40 studies has shown that a rational combination of two drugs from any two classes of antihypertensive agents significantly improves the degree of blood pressure reduction than increasing the dose of a single drug. Another advantage of combination therapy is that there may be physiological and pharmacological synergy between drugs from different classes, which not only leads to a significant decrease in blood pressure and good tolerability. Combination therapy also allows you to suppress counter-regulatory mechanisms of blood pressure increase. Rational combinations of antihypertensive drugs are ACE inhibitors + TD; BRA + TD; ACE inhibitor + AC; BRA + AK; dihydropyridine AC + BB; AK + TD; BB + TD [1].

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ORIGIN, DIAGNOSIS AND MODERN CLINICAL DIAGNOSTIC METHODS OF

HYPERTENSION

¹Uzoqova Oyjamol Narzullayevna

²Boboqulova Nilufar

³Axsanova Farida

¹Assistant Professor, Department of Hematology, Samarkand State Medical University

²'³Students of Samarkand State Medical University

https://doi.org/10.5281/zenodo.15023177

Relevance of the problem:

Many RCTs have shown that monotherapy reduces blood

pressure only in a limited number of hypertension cases, and most patients require a combination

of at least two drugs for satisfactory blood pressure control. A meta-analysis of more than 40

studies has shown that a rational combination of two drugs from any two classes of

antihypertensive agents significantly improves the degree of blood pressure reduction than

increasing the dose of a single drug. Another advantage of combination therapy is that there may

be physiological and pharmacological synergy between drugs from different classes, which not

only leads to a significant decrease in blood pressure and good tolerability. Combination therapy

also allows you to suppress counter-regulatory mechanisms of blood pressure increase. Rational

combinations of antihypertensive drugs are ACE inhibitors + TD; BRA + TD; ACE inhibitor +

AC; BRA + AK; dihydropyridine AC + BB; AK + TD; BB + TD [1].

Research methods and materials:

Taking into account the clinical course of the disease,

comorbid pathology, tolerability of treatment and side effect profile, as well as the presence of

benefits associated with the patient's personal positive or negative experience and, accordingly,

the expected adherence to treatment, the doctor has the right to prescribe any antihypertensive drug

registered in Russia, both in monotherapy and in combination therapy, if clinically appropriate. In

this case, deviations from standard treatment regimens require an appropriate explanation in the

anamnesis [1].

When the combination is not sufficiently effective, “stepping up” within the AHT

framework involves using higher doses of the combination or immediately switching to a 3-

component treatment regimen. Both approaches are acceptable in the phase of using a secondary

combination of antihypertensive agents, but they should ensure that the target blood pressure is

achieved within 3 months, with a dose titration phase of approximately 4 weeks [1].

When assessing the need for extended AHT, it should be borne in mind that target blood

pressure levels are recommended to be achieved in each subgroup of patients, but the most


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important principle for achieving them is to ensure safety and maintain the patient's quality of life.

Therefore, the speed of achieving target values and the degree of blood pressure reduction can be

adjusted for a particular patient depending on the specific clinical situation. In this case, poor

tolerance of blood pressure reduction may be a reason for a slower titration of doses and the

number of drugs prescribed; as with good tolerance to AHT, BP can be reduced to values lower

than the average recommended [1]. Failure to achieve target blood pressure within 3 months is not

considered AHT failure if this is associated with clinical necessity. If the physician considers that

poor compliance of the patient is an obstacle to achieving target BP, this should be reflected in the

medical record and measures should be taken and recorded to improve compliance. In such cases,

failure to achieve target levels should not be considered a failure of care [1]. Recommended

combinations of three antihypertensive drugs include ACE inhibitor + AC + diuretic and ARB +

AC + diuretic. Other combinations may be used, depending on the indication and in special

circumstances: ACE inhibitor + dihydropyridine AC + BB; BRA + dihydropyridine AC + BB;

ACE inhibitor + diuretic + BB; ARB + diuretic + BB; dihydropyridine AC + diuretic + beta-

blocker [1].

Low-dose aspirin (75–150 mg) is recommended for patients with hypertension and a

history of cardiovascular disease [1, 21]. Long-term use as part of secondary prevention reduces

cardiovascular mortality by 15% and nonfatal vascular events by 30% [1, 22]. In patients after MI,

acetylsalicylic acid use for 2 years is associated with an absolute reduction in the risk of

cardiovascular events of 33 ± 7% per 1000 patients treated within 1 month and 39 ± 5% per 1000

patients treated. After stroke or transient ischemic attack, the reduction in cardiovascular events is

27 ± 8% per 1000 patients treated for 34 months [1, 23]. In a study of patients with stable angina,

taking acetylsalicylic acid (75 mg daily) for 15 months compared with placebo reduced the overall

incidence of MI and sudden death by 34%, and other vascular events and cardiovascular death by

22–32% [1, 24].

Conclusions

: In 15–20% of patients, blood pressure control may not be achieved with three

drugs. In this case, a combination of ≥4 antihypertensive drugs (preferably in two tablets) is used.

However, in cases of resistant hypertension, the effectiveness of each new drug should be

monitored with the addition of their effect, and ineffective antihypertensive drugs should be

discontinued as part of a stepwise titration of multi-component AHT [1].

In case of intolerance to spironolactone, other diuretics (eplerenone, loop diuretics,

including high doses), beta-blockers, alpha-blockers, or centrally acting drugs can be used as the

4th component of hypertension therapy [1, 26].


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Eplerenone, like spironolactone, has shown positive effects in heart failure and resistant

hypertension. Spironolactone and eplerenone are used in the treatment of hypertension at low daily

doses (25–50 mg). Their use is absolutely contraindicated in patients with a creatinine clearance

<30 ml/min/1.73 m2, as this increases the risk of hyperkalemia and worsening renal function [1].

The imidazoline receptor agonist moxonidine increases tissue insulin sensitivity in

overweight patients with mild hypertension, insulin resistance, and impaired carbohydrate

metabolism. It is recommended for use in the treatment of patients with hypertension and

metabolic syndrome or obesity [1, 27]. In this group of patients, moxonidine may be considered

in combination with RAAS blockers (ACE inhibitors or ARBs), CA antagonists, or diuretics [1].

Conclusion

: According to the Eurasian Clinical Guidelines for the Prevention and

Treatment of Cardiovascular Disease in Patients with Diabetes and Prediabetes (2021), it is

recommended to consider the use of moxonidine + RAAS inhibitor (ACE inhibitor or ARB) + AC

or diuretics in patients with hypertension to control blood pressure: UUR - IIb, UDL - C [26]. We

should add that in patients with arterial hypertension with diabetes mellitus, it is recommended to

start antihypertensive therapy when the blood pressure measured in a medical institution is

≥140/90 mm Hg. The target blood pressure levels and the principles of stepwise therapy in this

case correspond to the hypertension treatment regimen presented in this material (Part I) [1, 26].

The use of moxonidine is contraindicated in cases of sick sinus syndrome, sinoatrial,

atrioventricular block 2-3 degrees, severe bradycardia with a heart rate <50 beats per minute, CHF

III-IV functional class [1].

The preferred indication for alpha-blockers (doxazosin, prazosin) is benign prostatic

hyperplasia in patients with hypertension. They improve carbohydrate and lipid metabolism,

increase tissue sensitivity to insulin, and improve renal hemodynamics. These drugs are used with

caution in patients with diabetic neuropathy and in patients over 65 years of age because they can

cause postural hypotension [1].

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2025

MARCH

NEW RENAISSANCE

INTERNATIONAL SCIENTIFIC AND PRACTICAL CONFERENCE

VOLUME 2

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ISSUE 3

115

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Sultanov S. et al. Long-term salbi effects of the covid-19 pandemic on the health of existing residents of alcohol addiction //Science and innovation. – 2023. – Т. 2. – №. D11. – С. 430-438.

Madaminov M., . Breast cancer detection methods, symptoms, causes, treatment //Science and innovation. – 2022. – Т. 1. – №. D8. – С. 530-535.

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Zhalalova D. et al. INFORMATION POINT OF PERIPHERAL BLOOD INDEXES IN THE DIAGNOSIS OF THE ETIOLOGY OF OPTIC NERVE DAMAGE //Science and innovation. – 2023. – Т. 2. – №. D11. – С. 124-130.

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Jalalova D., Raxmonov X., . ЗНАЧЕНИЕ ДИСФУНКЦИИ ЭНДОТЕЛИЯ В РАЗВИТИЕ РЕТИНОПАТИИ У БОЛЬНЫХ АГ И ПУТИ ЕГО КОРРЕКЦИИ //Science and innovation. – 2022. – Т. 1. – №. D8. – С. 101-113.

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Konstantinova, O., . (2023). Clinical and psychological characteristics of patients with alcoholism with suicidal behavior. Science and innovation, 2(D11), 399-404.

Qizi, T. J. I., . (2022). Treatment of myocardial infarction and first aid. Science and innovation, 1(D3), 317-320.

Xushvaktova D., . Clinical features of mental disorders in synthetic drug users //Science and innovation. – 2023. – Т. 2. – №. D10. – С. 242-247.

Solovyova Y. et al. The relevance of psychotic disorders in the acute period of a stroke //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 212-217.

Solovyova Y. et al. Suicide prevention in adolescents with mental disorders //Science and innovation. – 2023. – Т. 2. – №. D11. – С. 303-308.

Sultanov S. et al. Changes in alcohol behavior during the covid-19 pandemic and beyond //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 302-309.

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Hamidullayevna X. D., Temirpulatovich T. B. Factors of pathomorphosis of alcoholic delirium //Iqro jurnali. – 2023. – Т. 1. – №. 2. – С. 721-729.

Sharapova D. et al. Clinical and socio-economic effectiveness of injectable long-term forms of atypical antipsychotics in schizophrenia //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 290-295.

Sharapova D., . Psychological factors for the formation of aggressive behavior in the youth environment //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 404-408.

Ochilov U. et al. The question of the features of clinical and immunological parameters in the diagnosis of juvenile depression with" subpsychotic" symptoms //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 218-222.

Sharapova D., ., Turayev B. Prevalence of mental disorders in children and adolescents with cancer and methods of their treatment //Science and innovation. – 2023. – Т. 2. – №. D12. – С. 373-378.