Authors

  • Ibodillo Irgashev

DOI:

https://doi.org/10.71337/inlibrary.uz.science-research.69138

Keywords:

arterioscleros digoxin pulmonary oedema myocardial infarct antianginal effect cardiotonic effect isosorbide dinitrate.

Abstract

In economically developed countries, CVD accounts for 2.1% of the total population, with more than 90% of women and about 75% of men with CVD being patients over 70 years of age (V. A gv a ll e t a l., 1998). In Russia, the elderly include people aged 60 to 75 years, aged 75 to 90 years - people in old age and over 90 years - long-livers. In the USA and European countries the elderly include people aged 75-90 years (‘young elderly’), at the age of over 90 years - ‘old elderly’, long-livers.

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FEATURES AND BENEFITS OF CARDIAC GLYCOSIDES IN CHRONIC HEART

FAILURE

Irgashev Ibodillo Ergashevich

Faculty of Medicine, International University of Asia, Uzbekistan

Anesthesiologist-resuscitator.

https://doi.org/10.5281/zenodo.14911448

Abstract.

In economically developed countries, CVD accounts for 2.1% of the total

population, with more than 90% of women and about 75% of men with CVD being patients over

70 years of age (V. A gv a ll e t a l., 1998). In Russia, the elderly include people aged 60 to 75

years, aged 75 to 90 years - people in old age and over 90 years - long-livers. In the USA and

European countries the elderly include people aged 75-90 years (‘young elderly’), at the age of

over 90 years - ‘old elderly’, long-livers.

Keywords:

arterioscleros, digoxin, pulmonary oedema, myocardial infarct, antianginal

effect, cardiotonic effect, isosorbide dinitrate.

ОСОБЕННОСТИ И ПРЕИМУЩЕСТВА СЕРДЕЧНЫХ ГЛИКОЗИДОВ ПРИ

ХРОНИЧЕСКОЙ СЕРДЕЧНОЙ НЕДОСТАТОЧНОСТИ

Аннотация.

В экономически развитых странах ССЗ составляют 2,1% от общей

численности населения, при этом более 90% женщин и около 75% мужчин с ССЗ

являются пациентами старше 70 лет (В. Агвалл и др., 1998). В России к пожилым

относят людей в возрасте от 60 до 75 лет, в возрасте от 75 до 90 лет - людей в

старческом возрасте и старше 90 лет - долгожителей. В США и странах Европы к

пожилым относят людей в возрасте 75-90 лет («молодые пожилые»), в возрасте

старше 90 лет - «старые пожилые», долгожители.

Ключевые слова:

артериосклероз, дигоксин, отек легких, инфаркт миокарда,

антиангинальный эффект, кардиотонический эффект, изосорбида динитрат.

Increase in the frequency of CVD with age is caused by a number of significant factors:

undoubted growth in the modern world of CHD, AH - the main ‘suppliers’ of CVD,especially in

their frequent combination; certain successes in the treatment of acute and chronic forms of

CHD, BP, which contributed to the chronicisation of these diseases, increased life expectancy of

such patients with the development of circulatory decompensation. In addition, the increase in

the incidence of CVI with age is due to the formation of ‘senile heart’ with accumulation of

amyloid and lipofuscin in cardiomyocytes, sclerosis and atrophy of myocardium, increasing

processes of atherosclerosis not only of main arteries, but also arteriosclerosis, hyalinosis of


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small and smallest arteries and arterioles. Peripheral oedema in the elderly is not necessarily a

consequence of CVD.

They may be associated with increased tissue hydrophilicity, decreased colloid osmotic

pressure of blood, slow blood flow, decreased filtration capacity of the kidneys, varicose veins,

adynamia, chronic kidney disease, liver disease, etc. It should be especially noted the so-called

chronic left ventricular insufficiency with phenomena of incipient pulmonary oedema. These

conditions of recurrent cardiac asthma can stop independently, and sometimes require urgent

care. The presented features of CH in the elderly cause undoubted diagnostic difficulties, require

individualised treatment and motor rehabilitation. The peculiarities of treatment include:

- early administration of diuretics - from the initial stages of CH at first briefly, then

courses and combined;

- early use of peripheral vasodilators mainly nitrates, IAPPs, calcium antagonists;

- administration of cardiac glycosides for certain indications and in doses appropriate to

old age;

- if possible, sufficiently active motor rehabilitation.

Treatment of CHF in the elderly requires a number of additional conditions, taking into

account the considerable diagnostic difficulties and side effects of drug therapy.

It should be borne in mind that there are drugs that are not recommended for prescription

in CHF in the elderly. Theseinclude: non-steroidal anti-inflammatory drugs, corticosteroids, class

I antiarrhythmic drugs (quinidine, disopyramide, etacizine, etmosine, etc.).

Pharmacokinetics of cardiac glycosides in the elderly has its own peculiarities:

- increased absorption in the intestine due to weakened peristalsis and tendency to

constipation;

-increased content of active free fraction in blood plasma due to age-related albuminemia

and decreased amount of water in the div;

- slower excretion of glycosides by the kidneys and slower biotransformation in the liver

(this applies mainly to digoxin).

These features at the same dose of the drug provide the concentration of cardiac

glycosides in blood plasma in the elderly 1.5-2 times higher than in middle-aged people. Hence

the conclusion that in geriatric practice should be used reduced by 1.5-2 times doses of cardiac

glycosides. Pharmacodynamics of cardiac glycosides in old age also has certain peculiarities:

- increased sensitivity and decreased tolerance of myocardium to cardiac glycosides;

- more pronounced arrhythmogenic effect and greater refractoriness to the drugs.


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Age peculiarities of pharmacokinetics and pharmacodynamics determine not only the

severity of cardiotonic effect, but also the rapidity of glycoside intoxication. In this case, there is

a high threat of adverse events during glycoside therapy.

Cardiac glycosides (digoxin) in geriatric practice are prescribed in CVD only on strict

indications. After a few weeks, some patients become accustomed to nitrates. The effectiveness

of drugs is markedly reduced and, which is practically important, does not increase with

increasing single and daily doses.

Hemodynamic and antianginal effect of nitrates does not occur. In such cases, the doses

of nitrates should be gradually reduced until complete cancellation. After 1-2 weeks, sensitivity

to nitrates may be restored. It is possible to use mononitrates - olicard, monochinqué, etc., giving

less tolerance and greater haemodynamic effect.

Direct vasodilators (nitroglycerin and its derivatives, isosorbide dinitrate, mononitrates,

etc.) are widely used in the treatment of OSN (pulmonaryoedema, cardiogenic shock, etc.), as

well as in painful forms and other painless variants of chronic CHD in the elderly combined with

CVI. The use of the indicated drugs allows to achieve antianginal effect by reducing myocardial

ischaemia.

In recent years there appeared materials about cardioprotective effect of mononitrates

(olicard, monochinqué, etc.) in CVD. When they are administered with other cardiotropic drugs

(IAPP, cardiac glycosides, etc.), a significant improvement of the main haemodynamic

parameters in the treatment of CHF in the elderly was revealed.

Negative phenomena during the use of parenteral nitrates in the elderly occur in 40% of

observations and more often (acute headache, nausea, etc.). Headache is associated with venous

stasis, sharp arteriolodilatation of cerebral vessels. In case of severe headache it is possible to use

caffeine-benzoate sodium orally in the form of a solution (1 ampoule of caffeine solution per 5-7

ml of 40% glucose solution). Molsidomine also quite often (about 20% of cases) causes

headache, dizziness and nausea.

When hydralazine hydrochloride (apressin) isused in the elderly, headache, nausea and

vomiting, palpitations, hyperaemia of the skin, a feeling of heat and burning in the eyes

occurmore often than in middle-aged people.

The use of sodium nitroprusside and prazosin in the elderly, especially without detailed

clinical and haemodynamic control, may be accompanied by side effects in the form of

headache, nausea and vomiting, abdominal pain, hyperthermia, irritability, increased number of

angina attacks. ACE inhibitors are widely used in the therapy of CHF in elderly patients. They

have displaced in geriatric practice cardiac glycosides and peripheral vasodilators. Possible side

effects of IAPPs include skin rash, dry cough, loss of taste sensation, glomerulopathy


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(proteinuria), excessive arterial hypotension. When prescribing IAPP in the elderly, it is

necessary to exclude previous renal pathology (diffuse glomerulonephritis, pyelonephritis) in the

stage of CPN, careful titration of the drug dose to prevent uncontrolled arterial hypotension. It is

in the elderly with CHF it is advisable to use IAPPs with a distinct long-term, prolonged action,

not causing hypotension of the first dose. These include perindopril - 2-4 mg/day, quinapril - 2.5-

5 mg/day.

Administration of IAPP is reasonable in all classes of CHF, in left ventricular

dysfunction, not accompanied by symptoms of CHF. This is relevant for patients with

myocardial infarction with latent CH; they can be used with preserved LV systolic function,

preventing the development of overt CH and prolonging the period before decompensation. The

positive effect of IAPPs on heart rhythm disorders, atherogenesis, renal function, etc. has been

revealed.

A number of principlesshould be taken into accountwhen prescribing IAPPs forelderly

people with CHF: first of all, verified CH, absence of contraindications to the use of IAPPs;

special caution should be observed in case of CHF I V class according to NYHA, creatinine level

increase over 200 mmol/l, symptoms of generalised atherosclerosis. Treatment should be started

with minimal doses: captopril - 6.25 mg 3 times a day, enalapril - 2.5 mg 2 times, quinapril - 2.5

mg 2 times, perindopril - 2 mg 1 time. Doses are doubled every 3-7 days. If necessary, the

titration rate can be increased or decreased.

It should be emphasised that these arrhythmias may be an independent pathogenetic

factor in the development and exacerbation of CHF in the elderly. If drug treatment of life-

threatening arrhythmias isineffective, surgical treatment is possible - destruction (ablation) of the

bundle of Hiss, temporary and permanent electrical stimulation of the heart, implantation of

cardioverter-defibrillator.

Pharmacological correction of energy metabolism opens new perspectives in the

treatment of CH in the elderly. The use of cytoprotective drug trimetazidine in chronic CHD in

elderly with CHF is promising and pathogenetically justified. Anti-ischaemic, antianginal and

metabolic ffects of trimetazidine are confirmed in randomised controlled trials. Thedrug can be

used both as monotherapy and in combination with other known cardiotropic agents; in this case

an additive effectis observed, which is especially important in the treatment of CHD and CHF in

elderly people.


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Komilovich, E. B., & Jamshidovich, A. S. (2024). YURAK ISHEMIYASI. STENOKARDIYADA SHOSHILINCH TIBBIY YORDAM. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 12-20.

Komilovich, E. B., & Jamshidovich, A. S. (2024). HYPERTENSION ETIOLOGY. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 32-41.

Komilovich, E. B., & Jamshidovich, A. S. (2024). CARDIAC ISCHEMIA. ANGINA NURSING DIAGNOSIS AND CARE. Journal of new century innovations, 46(1), 44-52.

Jamshidovich, A. S. (2024). IMPORTANT INDICATIONS OF THE DRUG WOBENZYM. Journal of new century innovations, 46(1), 29-32.

Jamshidovich, A. S. (2024). THE RESULTS OF THE EFFECT OF THE DRUG VALIDOL. Journal of new century innovations, 46(1), 19-23.

Jamshidovich, A. S. (2024). VIFERON USE IN CHILDREN. Journal of new century innovations, 46(1), 24-28.

Jamshidovich, A. S. (2024). USE OF DUSPATALIN (MEBEVERINE HYDROCHLORIDE) IN GASTROINTESTINAL DISEASES. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(5), 93-97.

Jamshidovich, A. S. (2024). ЭФФЕКТЫ СИРОПА ДЕПАКИНА (ВАЛЬПРОЕВАЯ КИСЛОТА). Ta'lim innovatsiyasi va integratsiyasi, 14(2), 148-152.

Jamshidovich, A. S., & Komilovich, E. B. (2024). THE IMPORTANCE OF THE DRUG ALLOCHOL FOR CHRONIC CHOLECYSTITIS. Ta'lim innovatsiyasi va integratsiyasi, 14(2), 133-137.

Jamshidovich, A. S., & Komilovich, E. B. (2024). ВАЖНЫЕ СВОЙСТВА ПРЕПАРАТА ДЕ-НОЛ (субцитрат висмута). Ta'lim innovatsiyasi va integratsiyasi, 14(2), 143-147.

Jamshidovich, A. S., & Komilovich, E. B. (2024). SPECIAL FEATURES OF BUDECTON DRUG. Ta'lim innovatsiyasi va integratsiyasi, 14(2), 138-142.

Jamshidovich, A. S. (2024). ЭФФЕКТИВНОЕ ВОЗДЕЙСТВИЕ ПРЕПАРАТА КЕЙВЕР. Ta'lim innovatsiyasi va integratsiyasi, 15(3), 137-143.

Jamshidovich, A. S. (2024). USEFUL PROPERTIES OF THE DRUG YODOFOL. Ta'lim innovatsiyasi va integratsiyasi, 15(3), 144-149.

Jamshidovich, A. S. (2024). FITOTERAPIYANING AKUSHER-GINEKOLOGIYADA AHAMIYATI. Лучшие интеллектуальные исследования, 15(2), 121-125.

Jamshidovich, A. S. (2024). THE IMPORTANCE OF THE DRUG DOPROKIN. Лучшие интеллектуальные исследования, 15(2), 109-114.

Jamshidovich, A. S. (2024). THE EFFECT OF DOSTINEX ON THE BODY. Лучшие интеллектуальные исследования, 15(2), 115-120.

Jamshidovich, A. S. (2024). РЕЗУЛЬТАТЫ ЭФФЕКТИВНОГО ДЕЙСТВИЯ ПРЕПАРАТА КАНЕФРОН. Лучшие интеллектуальные исследования, 15(2), 138-143.

Jamshidovich, A. S. (2024). СОВРЕМЕННЫЕ ЭФФЕКТЫ ПРЕПАРАТА ИНДОЛ. Лучшие интеллектуальные исследования, 15(2), 126-131.

Jamshidovich, A. S. (2024). EFFECT OF ISMIZHEN DRUG ON BODY IMMUNITY. Лучшие интеллектуальные исследования, 15(2), 132-137.

Jamshidovich, A. S. (2024). POSITIVE EFFECTS OF THE DRUG CARCIL. Ta'lim innovatsiyasi va integratsiyasi, 15(3), 127-131.

Jamshidovich, A. S. (2024). PЕЗУЛЬТАТЫ ЭФФЕКТИВНОГО ДЕЙСТВИЯ KАВИНТОНА. Ta'lim innovatsiyasi va integratsiyasi, 15(3), 132-136.

Jamshidovich, A. S. (2024). Современный Эффект Спрея Мометазон. Research Journal of Trauma and Disability Studies, 3(3), 62-65.

Jamshidovich, A. S. (2024). THE ROLE OF" SIMONTE PLUS" DRUG IN THE MODERN TREATMENT OF BRONCHIAL ASTHMA. EUROPEAN JOURNAL OF MODERN MEDICINE AND PRACTICE, 4(5), 66-70.

Jamshidovich, A. S. (2024). FEATURES OF THE BIOMECHANISM OF THE DRUG LEVOMYCETIN (CHLORAMPHENICOL). EUROPEAN JOURNAL OF MODERN MEDICINE AND PRACTICE, 4(9), 298-301.

Jamshidovich, A. S. (2024). THE MOST IMPORTANT INDICATORS OF OMEGA 3 SUBSTANCE IN THE METABOLISM OF THE HUMAN BODY. EUROPEAN JOURNAL OF MODERN MEDICINE AND PRACTICE, 4(10), 113-117.

Komilovich, E. B., & Khalimovich, M. N. (2024). CARDIAC ISCHEMIA. ANGINA CLINICAL FORMS AND DIAGNOSIS. Journal of new century innovations, 46(1), 70-78.

Komilovich, E. B. (2024). CORONARY HEART DISEASE. ANGINA EMERGENCY CARE. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(7), 235-242.

Komilovich, E. B. (2024). YURAK ISHEMIK KASALLIGI. STENOKARDIYANI DAVOLASHNING ZAMONAVIY TAMOYILLARI. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 3-11.

Jamshidovich, A. S. (2024). THE MOST IMPORTANT BENEFITS OF GINGER FOR THE HUMAN BODY'S IMMUNITY. EUROPEAN JOURNAL OF MODERN MEDICINE AND PRACTICE, 4(11), 269-273.

Axmedov, S. (2024). THE SPECIFIC EFFECT OF THE DRUG" BAKLASAN" IN CEREBROVASCULAR DISEASES AND ITS PRACTICAL SIGNIFICANCE TODAY. Modern Science and Research, 3(12), 485-492.

Komilovich, E. B. Z. (2023). Coronary Artery Disease. EUROPEAN JOURNAL OF MODERN MEDICINE AND PRACTICE, 3(12), 81-87.

Komilovich, E. B. (2024). CORONARY HEART DISEASE. ANGINA TREATMENT. Journal of new century innovations, 46(1), 95-104.

Komilovich, E. B. (2024). HYPERTENSION TREATMENT. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(7), 227-234.

Эргашов, Б. К. (2024). ИШЕМИЧЕСКАЯ БОЛЕЗНЬ СЕРДЦА. СТЕНОКАРДИЯ ПРОФИЛАКТИКА. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 21-31.

Axmedov, S. (2025). ВАЖНЫЕ СВОЙСТВА ПРЕПАРАТА ЭСКУЗАН ПРИ СОСУДИСТЫХ ЗАБОЛЕВАНИЯХ. Modern Science and Research, 4(1), 380-387.

Эргашов, Б. К. (2024). ГИПЕРТОНИЧЕСКАЯ БОЛЕЗНЬ ДИАГНОСТИКА. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 70-78.

Komilovich, E. B. (2024). HYPERTENSION DIAGNOSTICS. ОБРАЗОВАНИЕ НАУКА И ИННОВАЦИОННЫЕ ИДЕИ В МИРЕ, 38(6), 42-49.

Axmedov, S. (2025). SPECIFIC PROPERTIES OF ROXERA DRUG IN CARDIOVASCULAR DISEASES. Modern Science and Research, 4(2), 472-479.

Xusenovich, M. S., & Turаpjаnovnа, Z. M. (2024). SEMIZLIKNING TURLI FENOTIPLARDA KARDIOMETABOLIK XAVF OMILLARINI TAQQOSLASH. SO ‘NGI ILMIY TADQIQOTLAR NAZARIYASI, 7(4), 112-116.

Husenovich, M. S., & Turabdjanovna, Z. M. (2024). STUDY OF DIURNAL PROFILE OF ARTERIAL HYPERTENSION IN DIFFERENT PHENOTYPE OBESITY. образование наука и инновационные идеи в мире, 43(1), 129-131.

Xusenovich, M. S. (2024, September). SEMIZLIKNI TURLI FENOTIPLARIDA YURAK QON-TOMIR KASALLIKLARINI KELIB CHIQISH XAVFI PROGNOZI. In INTERNATIONAL SCIENTIFIC RESEARCH CONFERENCE (Vol. 3, No. 26, pp. 15-18).

Xusenovich, M. S. (2024). O ‘ZBEKISTONDA RESPUBLIKASIDA YURAK-QON TOMIR KASALLIKLARI TARQALISHI VA HOZIRGI KUNDAGI KO’RILAYOTGAN CHORA TADBIRLAR. AMERICAN JOURNAL OF SOCIAL SCIENCE, 2(3), 79-82.

Xusenovich, M. S., & Allayarovich, A. A. (2024). O ‘ZBEKISTONDA YURAK-QON TOMIR KASALLIKLARI TARQALISHI VA HOZIRGI KUNDAGI TENDENSIYASI. MODELS AND METHODS FOR INCREASING THE EFFICIENCY OF INNOVATIVE RESEARCH, 4(38), 54-57.

Ravshanovna, X. L. (2021, June). MINIMALLY INVASIVE METHODS OF TREATMENT OF DENTAL CARIES IN ADULTS. In " ONLINE-CONFERENCES" PLATFORM (pp. 118-119).